丙酸睾酮/戊酸睾酮/十一烯酸睾酮 ,缩写为TP/TV/TUe ,以商品名Triolandren销售,是丙酸睾酮 (TP)、戊酸睾酮 (TV)和十一烯酸睾酮 (TUe)的注射 复方药物 ,全都是雄激素 /合成代谢类固醇 。[ 1] [ 2] [ 3] 它含有20mg/mL的TP、80mg/mL的TV和150mg/mL的TUe(总共250毫克的睾酮酯 和173.8毫克的游离睾酮 )油 溶液,并通过定期肌肉注射 给药。[ 1] [ 2] [ 3] [ 4] 据报道,该药物的作用持续时间约为10至20天。[ 1] [ 2]
^ 1.0 1.1 1.2 Schuermann H, Doepfmer R. Fertilitätsstörungen beim Manne . Springer-Verlag. 1960: 260–. ISBN 978-3-642-94784-1 .
^ 2.0 2.1 2.2 Ufer J. Hormontherapie in der Frauenheilkunde: Grundlagen und Praxis . Gruyter. 1960: 153. ISBN 9783111138770 .
^ 3.0 3.1 Aakvaag A, Vogt JH. Plasma testosterone values in different forms of testosterone treatment. Acta Endocrinologica. March 1969, 60 (3): 537–42. PMID 5395873 . doi:10.1530/acta.0.0600537 . Triolandren®, for intramuscular use, kindly supplied by Ciba, Basel, through Kobro 8c Co., Oslo, containing three different testosterone esters, in the following amounts of testosterone equivalents per ml oil: propionate 20 mg; valerate 80 mg; undecylenate 150 mg.
^ Zachmann M, Prader A. Anabolic and androgenic effect of testosterone in sexually immature boys and its dependency on growth hormone . The Journal of Clinical Endocrinology and Metabolism. January 1970, 30 (1): 85–95. PMID 4311616 . doi:10.1210/jcem-30-1-85 . Triolandren, CIBA; 250 mg of this preparation contains 20 mg of testosterone propionate, 80 mg of testosterone-n-valerianate, and 150 mg of testoster- one undecylenate—250 mg thus contains 173.8 mg of testosterone; the remaining 76.2 mg consists of the ester components [...]
激动药 抗雄激素
AR 受体拮抗剂 类固醇生成抑制剂
抗促性腺激素
D2 receptor antagonist s (prolactin releaser s) (e.g., domperidone , 甲氧氯普胺 , risperidone , haloperidol , 氯丙嗪 , sulpiride )
Estrogen s (e.g., bifluranol , 己烯雌酚 , 雌二醇 , estradiol ester s, ethinylestradiol , ethinylestradiol sulfonate , paroxypropione )
GnRH agonist s (e.g., leuprorelin )
GnRH antagonist s (e.g., cetrorelix )
Progestogen s (incl., chlormadinone acetate , 醋酸环丙孕酮 , hydroxyprogesterone caproate , gestonorone caproate , medroxyprogesterone acetate , megestrol acetate )
其它